Structure-based design of an N-terminal bromodomain selective BET inhibitor retaining the anti-inflammatory and antiproliferative phenotype

William Kerr, Christopher Wellaway

Research output: Contribution to conferenceSpeech

Original languageEnglish
Publication statusPublished - 25 Jun 2014
EventThe 8th WestCHEM Postgraduate Symposium in Organic Chemistry - University of Strathclyde, Glasgow, United Kingdom
Duration: 25 Jun 201425 Jun 2014

Conference

ConferenceThe 8th WestCHEM Postgraduate Symposium in Organic Chemistry
CountryUnited Kingdom
CityGlasgow
Period25/06/1425/06/14

Keywords

  • structure based design
  • bromodomain
  • BET inhibitors
  • extra-terminal proteins
  • anti-inflammatory
  • antiproliferative

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