Structure-based design of an N-terminal bromodomain selective BET inhibitor retaining the anti-inflammatory and antiproliferative phenotype

William Kerr, Christopher Wellaway

Research output: Contribution to conferenceSpeech

Conference

ConferenceThe 8th WestCHEM Postgraduate Symposium in Organic Chemistry
CountryUnited Kingdom
CityGlasgow
Period25/06/1425/06/14

Keywords

  • structure based design
  • bromodomain
  • BET inhibitors
  • extra-terminal proteins
  • anti-inflammatory
  • antiproliferative

Cite this

Kerr, W., & Wellaway, C. (2014). Structure-based design of an N-terminal bromodomain selective BET inhibitor retaining the anti-inflammatory and antiproliferative phenotype. The 8th WestCHEM Postgraduate Symposium in Organic Chemistry, Glasgow, United Kingdom.
Kerr, William ; Wellaway, Christopher. / Structure-based design of an N-terminal bromodomain selective BET inhibitor retaining the anti-inflammatory and antiproliferative phenotype. The 8th WestCHEM Postgraduate Symposium in Organic Chemistry, Glasgow, United Kingdom.
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title = "Structure-based design of an N-terminal bromodomain selective BET inhibitor retaining the anti-inflammatory and antiproliferative phenotype",
keywords = "structure based design, bromodomain, BET inhibitors, extra-terminal proteins, anti-inflammatory, antiproliferative",
author = "William Kerr and Christopher Wellaway",
year = "2014",
month = "6",
day = "25",
language = "English",
note = "The 8th WestCHEM Postgraduate Symposium in Organic Chemistry ; Conference date: 25-06-2014 Through 25-06-2014",

}

Kerr, W & Wellaway, C 2014, 'Structure-based design of an N-terminal bromodomain selective BET inhibitor retaining the anti-inflammatory and antiproliferative phenotype' The 8th WestCHEM Postgraduate Symposium in Organic Chemistry, Glasgow, United Kingdom, 25/06/14 - 25/06/14, .

Structure-based design of an N-terminal bromodomain selective BET inhibitor retaining the anti-inflammatory and antiproliferative phenotype. / Kerr, William; Wellaway, Christopher.

2014. The 8th WestCHEM Postgraduate Symposium in Organic Chemistry, Glasgow, United Kingdom.

Research output: Contribution to conferenceSpeech

TY - CONF

T1 - Structure-based design of an N-terminal bromodomain selective BET inhibitor retaining the anti-inflammatory and antiproliferative phenotype

AU - Kerr, William

AU - Wellaway, Christopher

PY - 2014/6/25

Y1 - 2014/6/25

KW - structure based design

KW - bromodomain

KW - BET inhibitors

KW - extra-terminal proteins

KW - anti-inflammatory

KW - antiproliferative

UR - http://www.westchem.ac.uk/

M3 - Speech

ER -

Kerr W, Wellaway C. Structure-based design of an N-terminal bromodomain selective BET inhibitor retaining the anti-inflammatory and antiproliferative phenotype. 2014. The 8th WestCHEM Postgraduate Symposium in Organic Chemistry, Glasgow, United Kingdom.