A preparatively accessible route to a series of conformationally-locked bicyclic morpholines has been developed. This flexible approach allows for diversification in order for a small array of lead-like scaffolds to be synthesised from readily available key building blocks.
|Number of pages||3|
|Journal||Journal of the Chemical Society, Chemical Communications|
|Early online date||15 Aug 2013|
|Publication status||Published - 10 Sept 2013|
- flexible access
- bicyclic morpholines