Craig Jamieson

Research output

Research output per year 2008 2020

• 44 Article
• 5 Patent
• 2 Chapter
• 1 Book
• 2 More
  • 1 Other chapter contribution
  • 1 Letter

Research output per year

Research output per year

Search results

• 2020

  A one-pot Suzuki-hydrogenolysis protocol for the modular synthesis of 2,5-diaryltetrazoles

  Livingstone, K., Bertrand, S. & Jamieson, C., 21 May 2020, In: Journal of Organic Chemistry. 85, 11, p. 7413-7423 11 p.

  Research output: Contribution to journal › Article › peer-review

  Open Access

  File

  • Hydrogenolysis
  • Photochemical reactions
  • Nitriles
  • Imines
  • Derivatives
  1 Citation (Scopus)

  6 Downloads (Pure)

• Design, synthesis and evaluation of E2-25K derived stapled peptides

  Watson, M. E., Scott, D., Jamieson, C., Layfield, R. & Mason, A. M., 24 Mar 2020, In: Peptide Science. 10 p., e24158.

  Research output: Contribution to journal › Article › peer-review

  Open Access

  File

  • Peptides
  • Proteins
  • Polyubiquitin
  • Ubiquitin-Conjugating Enzymes
  • Enzymes
  2 Downloads (Pure)

• Design and development of a macrocyclic series targeting phosphoinositide 3-kinase δ

  Spencer, J. A., Baldwin, I. R., Barton, N., Chung, C-W., Convery, M. A., Edwards, C. D., Jamieson, C., Mallett, D. N., Rowedder, J. E., Rowland, P., Thomas, D. A. & Hardy, C. J., 9 Jul 2020, In: ACS Medicinal Chemistry Letters . 11, 7, p. 1386-1391 6 p.

  Research output: Contribution to journal › Article › peer-review

  • Benzoxazines
  • Surface plasmon resonance
  • Pharmacokinetics
  • Solubility
  • Phosphatidylinositol 3-Kinase

• The Nitrile Imine 1,3-Dipole: Properties, Reactivity and Applications

  Jamieson, C. & Livingstone, K., 26 Mar 2020, Cham, Switzerland. 166 p.

  Research output: Book/Report › Book

  • Nitriles
  • Imines
  6 Citations (Scopus)

• Transition metal-free coupling of 1,3-dipoles and boronic acids as a sustainable approach to C-C bond formation

  Livingstone, K., Bertrand, S., Kennedy, A. R. & Jamieson, C., 17 Aug 2020, In: Chemistry - A European Journal. 26, 46, p. 10591-10597 7 p.

  Research output: Contribution to journal › Article › peer-review

  Open Access

  File

  • Boronic Acids
  • Nitriles
  • Transition metals
  • Imines
  • Oximes
  2 Citations (Scopus)

  9 Downloads (Pure)

• UV-induced 1,3,4-oxadiazole formation from 5-substituted tetrazoles and carboxylic acids in flow

  Green, L., Livingstone, K., Bertrand, S., Peace, S. & Jamieson, C., 20 Nov 2020, In: Chemistry - A European Journal. 26, 65, p. 14866-14870 5 p.

  Research output: Contribution to journal › Article › peer-review

  Open Access

  File

  • Tetrazoles
  • 1,3,4-oxadiazole
  • Carboxylic acids
  • Ultraviolet radiation
  • Carboxylic Acids
  1 Citation (Scopus)

  23 Downloads (Pure)
• 2019

  A fragment-like approach to PYCR1 inhibition

  Milne, K., Sun, J., Zaal, E. A., Mowat, J., Celie, P. H. N., Fish, A., Berkers, C. R., Forlani, G., Loayza-Puch, F., Jamieson, C. & Agami, R., 15 Sep 2019, In: Bioorganic and Medicinal Chemistry Letters . 29, 18, p. 2626-2631 6 p.

  Research output: Contribution to journal › Article › peer-review

  Open Access

  File

  • delta-1-pyrroline-5-carboxylate
  • Oxidoreductases
  • Proline
  • Pargyline
  • Biosynthesis
  4 Citations (Scopus)

  5 Downloads (Pure)

• A reappraisal of the Ni-[(Benzylprolyl)amino]benzophenone complex in the synthesis of α,α-disubstituted amino acid derivatives

  Watson, M. E., Jamieson, C., Kennedy, A. R. & Mason, A. M., 6 Sep 2019, In: Tetrahedron. 75, 36, 130485.

  Research output: Contribution to journal › Article › peer-review

  Open Access

  File

  • benzophenone
  • Derivatives
  • Amino Acids
  • Monomers
  • Proline
  3 Citations (Scopus)

  8 Downloads (Pure)

• Metal free C-C bond formation via coupling of nitrile imines and boronic acids

  Livingstone, K., Betrand, S., Mowat, J. & Jamieson, C., 28 Nov 2019, In: Chemical Science. 10, 44, p. 10412-10416 5 p.

  Research output: Contribution to journal › Article › peer-review

  Open Access

  File

  • Boronic Acids
  • Nitriles
  • Imines
  • Carbon
  • Metals
  7 Citations (Scopus)

  46 Downloads (Pure)

• Photocatalytic E→Z Isomerization of β-Ionyl Derivatives

  Livingstone, K., Tenberge, M., Pape, F., Daniliuc, C. G., Jamieson, C. & Gilmour, R., 6 Dec 2019, In: Organic Letters. 21, 23, p. 9677-9680 4 p.

  Research output: Contribution to journal › Article › peer-review

  Open Access

  File

  • Isomerization
  • Derivatives
  • Riboflavin
  • Isomers
  • Photocatalysts
  7 Citations (Scopus)

  4 Downloads (Pure)
• 2018

  Atom efficient synthesis of selectively difluorinated carbocycles through a gold(I) catalyzed cyclization

  McCarter, A. W., Sommer, M., Percy, J. M., Jamieson, C., Kennedy, A. R. & Hirst, D. J., 6 Jul 2018, In: Journal of Organic Chemistry.

  Research output: Contribution to journal › Article › peer-review

  Open Access

  File

  • Cyclization
  • Acetals
  • Atoms
  • Gold
  • Trifluoroethanol
  3 Citations (Scopus)

  5 Downloads (Pure)

• Cyrene as a bio-based solvent for HATU mediated amide coupling

  Wilson, K. L., Murray, J., Jamieson, C. & Watson, A. J. B., 28 Apr 2018, In: Organic and Biomolecular Chemistry. 16, p. 2851-2854 4 p.

  Research output: Contribution to journal › Article › peer-review

  Open Access

  File

  • Drug Discovery
  • Dipeptides
  • Peptides
  23 Citations (Scopus)

  15 Downloads (Pure)

• Scalable total synthesis and comprehensive structure–activity relationship studies of the phytotoxin coronatine

  Littleson, M. M., Baker, C. M., Dalencon, A. J., Frye, E. C., Jamieson, C., Kennedy, A. R., Ling, K. B., McLachlan, M. M., Montgomery, M. G., Russell, C. J. & Watson, A. J. B., 13 Feb 2018, (Accepted/In press) In: Nature Communications. 14 p.

  Research output: Contribution to journal › Article › peer-review

  Open Access

  File

  • coronafacic acid
  • coronatine
  • Agrochemicals
  • 1-amino-2-ethylcyclopropane-1-carboxylic acid
  • jasmonic acid
  72 Downloads (Pure)

• Surface functionalization with carboxylic acids by photochemical microcontact printing and tetrazole chemistry

  Buten, C., Lamping, S., Korsgen, M., Arlinghaus, H. F., Jamieson, C. & Ravoo, B. J., 16 Jan 2018, In: Langmuir. 17 p.

  Research output: Contribution to journal › Article › peer-review

  Open Access

  File

  • 1H-tetrazole
  • Carboxylic acids
  • Carboxylic Acids
  • Nucleophiles
  • Tetrazoles
  13 Citations (Scopus)

  97 Downloads (Pure)
• 2017

  Amidation of unactivated ester derivatives mediated by trifluoroethanol

  McPherson, C. G., Caldwell, N., Jamieson, C., Simpson, I. & Watson, A. J. B., 4 Apr 2017, In: Organic and Biomolecular Chemistry. 12 p.

  Research output: Contribution to journal › Article › peer-review

  Open Access

  File

  • Trifluoroethanol
  • Amines
  • Esters
  • Derivatives
  • Condensation
  20 Citations (Scopus)

  23 Downloads (Pure)

• A multicomponent route to functionalized amides and oxazolidinones

  McPherson, C. G., Cooper, A. K., Bubliauskas, A., Mulrainey, P., Jamieson, C. & Watson, A. J. B., 1 Dec 2017, In: Organic Letters. 4 p.

  Research output: Contribution to journal › Letter › peer-review

  Open Access

  File

  • Oxazolidinones
  • Epoxy Compounds
  • methyl carbonate
  • Esters
  • Oxindoles
  5 Citations (Scopus)

  17 Downloads (Pure)

• Emergence of small molecule non-RGD-mimetic inhibitors for RGD integrins

  Miller, L. M., Pritchard, J. M., Macdonald, S. J. F., Jamieson, C. & Watson, A. J. B., 30 Jan 2017, In: Journal of Medicinal Chemistry. 60, 8, 11 p.

  Research output: Contribution to journal › Article › peer-review

  Open Access

  File

  • Molecules
  • Integrins
  • Aspartic Acid
  • Ligands
  27 Citations (Scopus)

  98 Downloads (Pure)

• One-pot, three-step synthesis of cyclopropylboronic acid pinacol esters from synthetically tractable propargylic silyl ethers

  Spencer, J. A., Jamieson, C. & Talbot, E. P. A., 6 Jul 2017, In: Organic Letters. 4 p.

  Research output: Contribution to journal › Article › peer-review

  Open Access

  File

  • pinacol
  • Ethers
  • Esters
  • Lewis Acids
  • Cyclization
  13 Citations (Scopus)

  125 Downloads (Pure)

• Practical synthesis of pharmaceutically relevant molecules enriched in sp³ character

  Campbell, P. S., Jamieson, C., Simpson, I. & Watson, A. J. B., 27 Nov 2017, In: Chemical Communications (London). 4 p.

  Research output: Contribution to journal › Article › peer-review

  Open Access

  File

  • Molecules
  • Bioactivity
  • Drug Discovery
  • Hydrogenation
  10 Citations (Scopus)

  14 Downloads (Pure)

• Rational design of autotaxin inhibitors by structural evolution of endogenous modulators

  Keune, W-J., Potjewyd, F., Heidebrecht, T., Salgado-Polo, F., Macdonald, S. J. F., Chelvarajan, L., Abdel Latif, A., Soman, S., Morris, A. J., Watson, A. J. B., Jamieson, C. & Perrakis, A., 9 Mar 2017, In: Journal of Medicinal Chemistry. 60, 5, p. 2006-2017 12 p.

  Research output: Contribution to journal › Article › peer-review

  Open Access

  File
  14 Citations (Scopus)

  25 Downloads (Pure)

• Structure-activity relationships of small molecule autotaxin inhibitors with a discrete binding mode

  Miller, L. M., Keune, W-J., Castagna, D., Young, L. C., Duffy, E. L., Potjewyd, F., Salgado-Polo, F., Garcia, P. E., Semaan, D., Pritchard, J. M., Perrakis, A., Macdonald, S. J. F., Jamieson, C. & Watson, A. J. B., 26 Jan 2017, In: Journal of Medicinal Chemistry. 60, 2, p. 722-748 27 p.

  Research output: Contribution to journal › Article › peer-review

  Open Access

  File
  17 Citations (Scopus)

  73 Downloads (Pure)
• 2016

  Evolution of a novel orally bioavailable series of PI3Kδ inhibitors from an inhaled lead for the treatment of respiratory disease.

  Amour, A., Barton, N., Cooper, A. W. J., Inglis, G., Jamieson, C., Luscombe, C. N., Perez, D., Peace, S., Rowland, P., Tame, C., Uddin, S., Vitulli, G. & Wellaway, N., 18 Jul 2016, In: Journal of Medicinal Chemistry. 34 p.

  Research output: Contribution to journal › Article › peer-review

  Open Access

  File
  19 Citations (Scopus)

  72 Downloads (Pure)

• Investigation of a bicyclo[1.1.1]pentane as a phenyl replacement within an LpPLA2 inhibitor

  Measom, N., Down, K. D., Hirst, D. J., Jamieson, C., Manas, E. S., Patel, V. K. & Somers, D. O., 15 Nov 2016, In: ACS Medicinal Chemistry Letters . 7, 6 p.

  Research output: Contribution to journal › Article › peer-review

  Open Access

  File

  • dichlorocarbene
  • pentane
  • butane
  • X rays
  51 Citations (Scopus)

  82 Downloads (Pure)

• Palladium-catalyzed synthesis of aryl amides through silanoate-mediated hydrolysis of nitriles

  McPherson, C. G., Livingstone, K., Jamieson, C. & Simpson, I., 4 Jan 2016, In: Synlett. 27, 1, p. 88-92 5 p.

  Research output: Contribution to journal › Article › peer-review

  Open Access

  File

  • Imidoesters
  • Nitriles
  • Palladium
  • Bromides
  • Hydrolysis
  6 Citations (Scopus)

  51 Downloads (Pure)

• Scope and limitations of a DMF bio-alternative within Sonogashira cross-coupling and Cacchi-type annulation

  Wilson, K., Kennedy, A., Murray, J., Greatex, B., Jamieson, C. & Watson, A., 8 Sep 2016, In: Beilstein Journal of Organic Chemistry . 12, p. 2005-2011 7 p.

  Research output: Contribution to journal › Article › peer-review

  Open Access

  File

  • Agrochemicals
  • Industry
  • Pharmaceutical Preparations
  40 Citations (Scopus)

  379 Downloads (Pure)

• Structurally diverse mitochondrial branched chain aminotransferase (BCATm) leads with varying binding modes identified by fragment screening

  Borthwick, J. A., Ancellin, N., Bertrand, S. M., Bingham, R. P., Carter, P. S., Chung, C., Churcher, I., Dodic, N., Fournier, C., Francis, P. L., Hobbs, A., Jamieson, C., Pickett, S. D., Smith, S. E., Somers, D. ON., Spitzfaden, C., Suckling, C. J. & Young, R. J., 24 Mar 2016, In: Journal of Medicinal Chemistry. 59, 6, p. 2452-2467 16 p.

  Research output: Contribution to journal › Article › peer-review

  Open Access

  File

  • branched-chain-amino-acid transaminase
  • Screening
  • X ray crystallography
  • Nuclear magnetic resonance
  • Assays
  12 Citations (Scopus)

  57 Downloads (Pure)

• Synthetic approaches to coronafacic acid, coronamic acid, and coronatine

  Littleson, M. M., Russell, C. J., Frye, E. C., Ling, K. B., Jamieson, C. & Watson, A. J. B., 15 Aug 2016, In: Synthesis. 48, 20 p.

  Research output: Contribution to journal › Article › peer-review

  Open Access

  File

  • coronafacic acid
  • 1-amino-2-ethylcyclopropane-1-carboxylic acid
  • coronatine
  • Acids
  • Plant Growth Regulators
  5 Citations (Scopus)

  154 Downloads (Pure)
• 2015

  Catalytic amidation of unactivated ester derivatives mediated by trifluoroethanol

  Caldwell, N., Jamieson, C., Simpson, I. & Watson, A. J. B., 11 Jun 2015, In: Chemical Communications. 51, 46, p. 9495-9498 4 p.

  Research output: Contribution to journal › Article › peer-review

  Open Access

  File

  • Trifluoroethanol
  • Esters
  • Derivatives
  • Amides
  • Amines
  39 Citations (Scopus)

  44 Downloads (Pure)

• Identification of a novel class of autotaxin inhibitors through cross-screening

  Castagna, D., Duffy, E. L., Semaan, D., Young, L. C., Pritchard, J. M., Macdonald, S. J. F., Budd, D. C., Jamieson, C. & Watson, A. J. B., 1 Jun 2015, In: MedChemComm. 2015, 6, p. 1149-1155 6 p.

  Research output: Contribution to journal › Article › peer-review

  Open Access

  File

  • Lead compounds
  • Lysophosphatidic Acid Receptors
  • lysophosphatidic acid
  • Solubility
  • Screening
  8 Citations (Scopus)

  78 Downloads (Pure)

• Rational design of a novel AMPA receptor modulator through a hybridization approach

  Caldwell, N., Harms, J. E., Partin, K. M. & Jamieson, C., 2015, In: ACS Medicinal Chemistry Letters .

  Research output: Contribution to journal › Article › peer-review

  Open Access

  File

  • AMPA Receptors
  • Modulators
  • Ligands
  • Crystal structure
  • Ion Channels
  8 Citations (Scopus)

  100 Downloads (Pure)

• The discovery of in vivo active mitochondrial branched-chain aminotransferase (BCATm) inhibitors by hybridizing fragment and HTS hits

  Bertrand, S. M., Ancellin, N., Beaufils, B., Bingham, R. P., Borthwick, J. A., Boullay, A. B., Boursier, E., Carter, P. S., Chung, C. W., Churcher, I., Dodic, N., Fouchet, M. H., Fournier, C., Francis, P. L., Gummer, L. A., Herry, K., Hobbs, A., Hobbs, C. I., Homes, P., Jamieson, C. & 12 others, Nicodeme, E., Pickett, S. D., Reid, I. H., Simpson, G. L., Sloan, L. A., Smith, S. E., Somers, D. O. N., Spitzfaden, C., Suckling, C. J., Valko, K., Washio, Y. & Young, R. J., 24 Sep 2015, In: Journal of Medicinal Chemistry. 58, 18, p. 7140-7163 24 p.

  Research output: Contribution to journal › Article › peer-review

  • branched-chain-amino-acid transaminase
  • Pyrimidinones
  • Pharmacokinetics
  • Branched Chain Amino Acids
  • Physicochemical properties
  20 Citations (Scopus)
• 2014

  Amidation of esters with amino alcohols using organobase catalysis

  Caldwell, N., Campbell, P. S., Jamieson, C., Potjewyd, F., Simpson, I. & Watson, A. J. B., 3 Oct 2014, In: Journal of Organic Chemistry. 79, 19, p. 9347-9354 8 p.

  Research output: Contribution to journal › Article › peer-review

  Open Access

  File

  • methyl carbonate
  • Amino Alcohols
  • Oxazolidinones
  • Catalysis
  • Transesterification
  26 Citations (Scopus)

  129 Downloads (Pure)

• Molar efficiency: a useful metric to gauge relative reaction efficiency in discovery medicinal chemistry

  McGonagle, F. I., Sneddon, H. F., Jamieson, C. & Watson, A., 3 Mar 2014, In: ACS Sustainable Chemistry and Engineering. 2, 3, p. 523-532 10 p.

  Research output: Contribution to journal › Article › peer-review

  • Pharmaceutical Chemistry
  • Gages
  28 Citations (Scopus)

• Regiospecific synthesis of N2-aryl 1,2,3-triazoles from 2,5-disubstituted tetrazoles via photochemically generated nitrile imine intermediates

  Stewart, S., Harris, R. & Jamieson, C., 2014, In: Synlett. 25, 17, p. 2480-2484 5 p.

  Research output: Contribution to journal › Article › peer-review

  Open Access

  File

  • Tetrazoles
  • Nitriles
  • Imines
  • Triazoles
  • Derivatives
  9 Citations (Scopus)

  170 Downloads (Pure)
• 2013

  Development of a solvent selection guide for aldehyde-based direct reductive amination processes

  McGonagle, F. I., MacMillan, D. S., Murray, J., Sneddon, H. F., Jamieson, C. & Watson, A. J. B., 1 May 2013, In: Green Chemistry. 15, 5, p. 1159-1165 7 p.

  Research output: Contribution to journal › Article › peer-review

  • Amination
  • Aldehydes
  • Reducing Agents
  45 Citations (Scopus)

• Development of a sustainable catalytic ester amidation process

  Caldwell, N., Jamieson, C., Simpson, I. & Watson, A. J. B., 7 Oct 2013, In: ACS Sustainable Chemistry and Engineering. 1, 10, p. 1339-1344 6 p.

  Research output: Contribution to journal › Article › peer-review

  Open Access

  File

  • Esters
  • Amino alcohols
  • Amino Alcohols
  • Derivatives
  • 1-Propanol
  29 Citations (Scopus)

  85 Downloads (Pure)

• Evaluation of alternative solvents in common amide coupling reactions: replacement of dichloromethane and N,N-dimethylformamide

  MacMillan, D., Murray, J., Sneddon, H. F., Jamieson, C. & Watson, A., 2013, In: Green Chemistry. 15, 3, p. 596-600 5 p.

  Research output: Contribution to journal › Article › peer-review

  Open Access

  File

  • Dimethylformamide
  • Dichloromethane
  • Amides
  • Methylene Chloride
  91 Citations (Scopus)

  254 Downloads (Pure)

• Functional analysis of a novel positive allosteric modulator of AMPA receptors derived from a structure-based drug design strategy

  Harms, J. E., Benveniste, M., Maclean, J. K. F., Partin, K. M. & Jamieson, C., Jan 2013, In: Neuropharmacology. 64, p. 45-52 8 p.

  Research output: Contribution to journal › Article › peer-review
  23 Citations (Scopus)

• Organobase-catalyzed amidation of esters with amino alcohols

  Caldwell, N., Jamieson, C., Simpson, I. & Tuttle, T., 17 May 2013, In: Organic Letters. 15, 10, p. 2506-2509 4 p.

  Research output: Contribution to journal › Article › peer-review

  • Amino Alcohols
  • Esters
  35 Citations (Scopus)
• 2012

  AMPA receptor positive modulators

  Jamieson, C., Morrow, J. & Maclean, J., Jul 2012, Targets and Emerging Therapies for Schizophrenia. Albert, J. & Wood, M. (eds.). 1 ed. Hoboken, NJ, p. 187-231 44 p.

  Research output: Chapter in Book/Report/Conference proceeding › Chapter

• Replacement of dichloromethane within chromatographic purification: a guide to alternative solvents

  MacMillan, D. S., Murray, J., Sneddon, H. F., Jamieson, C. & Watson, A., 2012, In: Green Chemistry. 14, 11, p. 3016-3019 4 p.

  Research output: Contribution to journal › Article › peer-review

  Open Access

  File

  • Pharmaceutical Chemistry
  • Dichloromethane
  • Methylene Chloride
  • Purification
  • Molecules
  36 Citations (Scopus)

  403 Downloads (Pure)
• 2011

  Amino-heteroaryl derivatives as HCN blockers

  Grove, S. J. A., Morrison, A. J., Jamieson, C., Palin, R. & Maclean, J. K. F., 30 Jun 2011, IPC No. PCT/EP2010/070213, Patent No. WO2011076723A1

  Research output: Patent

  • 3-fluorophenol
  • Salts
  • Derivatives
  • Guanidine
  • Hydrolysis

• Structure based evolution of a novel series of positive modulators of the AMPA receptor

  Jamieson, C., Maclean, J. K. F., Brown, C. I., Campbell, R. A., Gillen, K. J., Gillespie, J., Kazemier, B., Kiczun, M., LAMONT, YVONNE., Lyons, A. J., Moir, E. M., Morrow, J. A., Pantling, J., Rankovic, Z. & Smith, L., 15 Jan 2011, In: Bioorganic and Medicinal Chemistry Letters. 21, 2, p. 805-811 7 p.

  Research output: Contribution to journal › Article › peer-review

  Open Access

  File

  • AMPA Receptors
  • Modulators
  26 Citations (Scopus)

  103 Downloads (Pure)
• 2010

  A novel series of positive modulators of the AMPA receptor: structure-based lead optimization

  Jamieson, C., Campbell, R. A., Cumming, I. A., Gillen, K. J., Gillespie, J., Kazemier, B., Kiczun, M., Lamont, Y., Lyons, A. J., Maclean, J. K. F., Martin, F., Moir, E. M., Morrow, J. A., Pantling, J., Rankovic, Z. & Smith, L., 15 Oct 2010, In: Bioorganic and Medicinal Chemistry Letters. 20, 20, p. 6072-6075 4 p.

  Research output: Contribution to journal › Article › peer-review

  Open Access

  File

  • Biological Availability
  • AMPA Receptors
  • Modulators
  • Lead compounds
  • X rays
  23 Citations (Scopus)

  283 Downloads (Pure)

• A novel series of positive modulators of the AMPA receptor: discovery and structure based hit-to-lead studies

  Jamieson, C., Basten, S., Campbell, R. A., Cumming, I. A., Gillen, K. J., Gillespie, J., Kazemier, B., Kiczun, M., Lamont, Y., Lyons, A. J., Maclean, J. K. F., Moir, E. M., Morrow, J. A., Papakosta, M., Rankovic, Z. & Smith, L., 1 Oct 2010, In: Bioorganic and Medicinal Chemistry Letters. 20, 19, p. 5753-5756 4 p.

  Research output: Contribution to journal › Article › peer-review

  Open Access

  File

  • AMPA Receptors
  • Modulators
  • Glutamate Receptors
  • Demonstrations
  • Pharmaceutical Preparations
  31 Citations (Scopus)

  86 Downloads (Pure)

• Dioxo-triazines as a novel series of cathepsin K inhibitors

  Rankovic, Z., Cai, J., Fradera, X., Dempster, M., Mistry, A., Long, C., Hamilton, E., King, A., Boucharens, S., Jamieson, C., Gillespie, J., Cumming, I., Uitdehaag, J. & van Zeeland, M., 1 Mar 2010, In: Bioorganic and Medicinal Chemistry Letters. 20, 5, p. 1488-1490 3 p.

  Research output: Contribution to journal › Article › peer-review

  • Triazines
  • Cathepsin K
  • Assays
  14 Citations (Scopus)

• High throughput screening approach to lead discovery

  Rankovic, Z., Jamieson, C. & Morphy, R., 2010, Lead Generation Approaches in Drug Discovery. Hoboken, NJ, p. 21-71 51 p.

  Research output: Chapter in Book/Report/Conference proceeding › Other chapter contribution

  7 Citations (Scopus)

• Positive allosteric modulators of the a-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid (AMPA) receptor

  Grove, S. J. A., Jamieson, C., Maclean, J. K. F., Morrow, J. A. & Rankovic, Z., 2010, In: Journal of Medicinal Chemistry. 53, 20, p. 7271-7279 8 p.

  Research output: Contribution to journal › Article › peer-review

  Open Access

  File
  29 Citations (Scopus)

  231 Downloads (Pure)

• Preparation of indane derivatives for treating and preventing psychiatric diseases.

  Gillen, K. J., Gillespie, J., Jamieson, C., MacLean, J. K. F., Moir, E. M. & Rankovic, Z., 14 Oct 2010, Patent No. WO2010115952A1

  Research output: Patent

  • Psychiatry
  • AMPA Receptors
  • Patents and inventions
  • 2-aminoindan
  • alkoxyl radical
• 2009

  Heterocyclic derivatives.

  Gallagher, M. G., Jamieson, C. C., Lyons, A. J., MacLean, J. K. F. & Moir, E. M., 21 May 2009, Patent No. US20090131455A1

  Research output: Patent